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Titel |
TI |
[EN] ALBICIDIN DERIVATIVES, THEIR USE AND SYNTHESIS
[FR] DÉRIVÉS D'ALBICIDINE, LEUR UTILISATION ET LEUR SYNTHÈSE |
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Anmelder/Inhaber |
PA |
CIRAD, FR
;
UNIV BERLIN TECH, DE
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| 72 |
Erfinder |
IN |
COCIANCICH STÉPHANE, FR
;
GRÄTZ STEFAN, DE
;
HÜGELLAND MANUELA, DE
;
KERWAT DENNIS, DE
;
KRETZ JULIAN, DE
;
PESIC ALEXANDER, DE
;
ROTT PHILLIPE, FR
;
ROYER MONIQUE, FR
;
SCHUBERT VIVIEN, DE
;
SÜSSMUTH RODERICH, DE
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Anmeldedatum |
AD |
14.02.2014 |
| 21 |
Anmeldenummer |
AN |
2014052922 |
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Anmeldeland |
AC |
EP |
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Veröffentlichungsdatum |
PUB |
21.08.2014 |
33
31
32 |
Priorität |
PRC
PRN
PRD |
EP
13170957
06.06.2013
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33
31
32 |
PRC
PRN
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EP
13192247
08.11.2013
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33
31
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EP
13199920
31.12.2013
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33
31
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PRD |
EP
13199921
31.12.2013
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33
31
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PRN
PRD |
EP
13199922
31.12.2013
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33
31
32 |
PRC
PRN
PRD |
US
201361765056
15.02.2013
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| 51 |
IPC-Hauptklasse |
ICM |
C07C 255/57
(2006.01)
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| 51 |
IPC-Nebenklasse |
ICS |
A61K 31/277
(2006.01)
A61K 31/5375
(2006.01)
A61P 31/04
(2006.01)
C07C 233/83
(2006.01)
C07C 255/03
(2006.01)
C07C 311/21
(2006.01)
C07D 207/34
(2006.01)
C07D 241/28
(2006.01)
C07D 277/56
(2006.01)
C07D 295/14
(2006.01)
C07D 307/56
(2006.01)
C07D 317/08
(2006.01)
C07D 333/38
(2006.01)
C07F 9/09
(2006.01)
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ICA |
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IPC-Indexklasse |
ICI |
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Gemeinsame Patentklassifikation |
CPC |
A61P 31/04
A61P 31/06
C07C 233/83
C07C 237/42
C07C 255/03
C07C 255/29
C07C 255/44
C07C 255/57
C07C 2601/02
C07C 2601/08
C07C 2601/14
C07C 2601/18
C07C 2603/74
C07C 275/42
C07C 311/21
C07C 311/46
C07C 311/47
C07D 207/34
C07D 209/34
C07D 213/81
C07D 237/24
C07D 241/24
C07D 263/24
C07D 277/56
C07D 295/14
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C07D 307/56
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C07D 317/08
C07D 317/46
C07D 333/38
C07F 9/062
C07F 9/09
C07F 9/12
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MCD-Hauptklasse |
MCM |
C07C 255/57
(2006.01)
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MCD-Nebenklasse |
MCS |
A61K 31/277
(2006.01)
A61K 31/5375
(2006.01)
A61P 31/04
(2006.01)
C07C 233/83
(2006.01)
C07C 255/03
(2006.01)
C07C 311/21
(2006.01)
C07D 207/34
(2006.01)
C07D 241/28
(2006.01)
C07D 277/56
(2006.01)
C07D 295/14
(2006.01)
C07D 307/56
(2006.01)
C07D 317/08
(2006.01)
C07D 333/38
(2006.01)
C07F 9/09
(2006.01)
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| 57 |
Zusammenfassung |
AB |
[EN] The present invention relates to a antibiotically active compounds characterized by general formula (I), wherein X1, BB, BC, BD, BE and X2 are building blocks with D1, D2, D3, D4 or D5 being linkers which comprise carbon, sulphur, nitrogen, phosphor and/or oxygen atoms and which are covalently connecting the moities BA and BB, BB and BC, BC and BD, BD and BE and BE and BF, respectively, and wherein in particular the building block BC comprises an amino acid derivative. The invention relates further to said compounds for use in a method of treatment of diseases, in particular for use in a method of treatment of bacterial infections.
[FR] La présente invention concerne des composés actifs sur le plan antibiotique caractérisés par la formule générale (I), dans laquelle X1, BB, BC, BD, BE et X2 sont des synthons, D1, D2, D3, D4 ou D5 étant des lieurs qui comprennent des atomes de carbone, de soufre, d'azote, de phosphore et/ou d'oxygène et qui raccordent de manière covalente les fractions BA et BB, BB et BC, BC et BD, BD et BE et BE et BF, respectivement, et le synthon BC comprenant en particulier un dérivé d'acide aminé. L'invention concerne en outre lesdits composés pour leur utilisation dans un procédé de traitement de maladies, en particulier pour leur utilisation dans un procédé de traitement d'infections bactériennes. |
| 56 |
Entgegengehaltene Patentdokumente/Zitate,
in Recherche ermittelt |
CT |
US000004525354A
US020110178104A1
WO002004035760A2
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| 56 |
Entgegengehaltene Patentdokumente/Zitate,
vom Anmelder genannt |
CT |
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| 56 |
Entgegengehaltene Nichtpatentliteratur/Zitate,
in Recherche ermittelt |
CTNP |
DATABASE CAPLUS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; KAI, AKIYOSHI ET AL: "Preparation of benzamides as insecticides for agriculture and gardening", XP002727098, retrieved from STN Database accession no. 2006:1174191 7;
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